Organic Chemistry

Alcohol, Phenol and Ethers

Preparation, Properties & Reactions of Hydroxy Compounds & Ethers

High Weightage in JEE Main & NEET

Introduction to Alcohols, Phenols & Ethers

Hydroxy compounds have -OH group attached to aliphatic or aromatic carbon. Alcohols are classified as monohydric, dihydric, trihydric based on number of -OH groups.

Alcohols: R-OH; Phenols: Ar-OH; Ethers: R-O-R'.

Classification of Alcohols

Monohydric (1°/2°/3°), Dihydric (Glycols), Trihydric (Glycerol).

Preparation of Monohydric Alcohols

From Alkyl Halides

RX + Aq. KOH → ROH + KX

1° halides give good yield; 3° give alkenes.

From Alkenes

Hydration
Direct: H2SO4/H2O (Markovnikov)
Oxymercuration: Hg(OAc)2/H2O, NaBH4
Hydroboration: BH3, H2O2/NaOH (Anti-Markovnikov)

From Carbonyl Compounds

Compound Reagent Product
Aldehyde (RCHO)LiAlH4 or H2/Pd1° Alcohol (RCH2OH)
Ketone (RCOR')NaBH4 or LiAlH42° Alcohol (RCH(OH)R')
Carboxylic Acid (RCOOH)LiAlH41° Alcohol (RCH2OH)
Ester (RCOOR')LiAlH4RCH2OH + R'OH

From Grignard Reagents

RMgX + HCHO → RCH2OMgX → RCH2OH (1°)
RMgX + R'CHO → RR'CHOMgX → RR'CHOH (2°)
RMgX + R'COR'' → RR'R''COMgX → RR'R''COH (3°)

Industrial Methods

Oxo Process: Alkene + CO + H2 → Aldehyde → Alcohol

Physical Properties of Alcohols

Solubility & BP
Lower alcohols miscible in water due to H-bonding
Solubility: 1° > 2° > 3°; Decreases with size
BP higher than alkanes/ethers due to H-bonding
BP: 1° > 2° > 3°
Other
Neutral, lower are liquids, higher solids
Methanol toxic, ethanol intoxicating

Chemical Properties of Alcohols

Acidity & O-H Cleavage

Alcohols weak acids: ROH + Na → RONa + 1/2H2

Acidity: 1° > 2° > 3°

Esterification: ROH + R'COOH → R'COOR + H2O

C-O Cleavage

With HX
ROH + HX → RX + H2O (Reactivity: HI > HBr > HCl; 3° > 2° > 1°)
With PCl5/PCl3/SOCl2
ROH + PCl5 → RCl + POCl3 + HCl
SOCl2 + Pyridine: Retention/Inversion

Dehydration

ROH → Alkene + H2O (H2SO4, ; 3° > 2° > 1°; Saytzeff rule)

Oxidation

Alcohol Type Product Reagent
Aldehyde/Carboxylic AcidPCC/K2Cr2O7
KetoneK2Cr2O7
No Reaction-

Distinction Tests

Test
Lucas (ZnCl2/HCl)No Rx/Heat5 minImmediate
Victor MeyerRedBlueNo Colour
IodoformCH3CH(OH)RCH3CORCH3C(OH)R2

Polyhydric Alcohols

Dihydric (Ethylene Glycol)

Preparation: From Ethylene, Dibromoethane

Properties: Colourless, viscous, antifreeze

Reactions: Esterification, Dehydration to Aldehydes

Trihydric (Glycerol)

Preparation: From Oils/Fats, Propene

Properties: Colourless, viscous, hygroscopic

Reactions: Nitration to Nitroglycerin, Oxidation

Uses: Explosives, Antifreeze, Soaps

Phenols

Preparation

Methods
From Haloarenes (Dow)
From Diazonium Salts
From Cumene (Industrial)
From Sulphonic Acid

Physical Properties

Colourless solid/liquid, characteristic smell, soluble in water due to H-bonding, higher BP than hydrocarbons.

Chemical Properties

Stronger acid than alcohols: Forms phenoxide

C6H5OH + Na → C6H5ONa + 1/2H2

Electrophilic Substitution: Ortho/Para directing, Halogenation, Nitration, Reimer-Tiemann (CHO), Kolbe (COOH)

Other: Esterification, Ether formation, Oxidation to Quinone

Tests

FeCl3: Violet; Br2 water: White ppt; Liebermann: Green/Blue

Derivatives of Phenol

Compound Preparation Properties/Uses
Picric AcidPhenol + Conc HNO3Yellow explosive, dye
CatecholFrom o-Phenolsulphonic AcidDeveloper, Antioxidant
ResorcinolFrom m-Benzenedisulphonic AcidAntiseptic, Dyes
HydroquinoneFrom p-BenzoquinoneDeveloper, Antioxidant

Ethers

Preparation

Williamson: RX + R'ONa → ROR'

Dehydration: 2ROH → ROR + H2O (H2SO4, 140°C)

From Alkyl Halides + Ag2O

Physical Properties

Gases/Liquids, low BP, soluble in water like alcohols, dipole moment.

Chemical Properties

Peroxide Formation, Hydrolysis with HI/HBr, Halogenation

Ring Substitution in Aromatic Ethers (o/p directing)

Important Points for Exams

High Yield Concepts

  • Preparation Methods: Grignard, Hydroboration (Anti-Markovnikov)
  • Oxidation: 1° → Aldehyde/Acid, 2° → Ketone, 3° No Rx
  • Dehydration: Saytzeff Rule, 3° > 2° > 1°
  • Phenol Acidity & Reactions: Reimer-Tiemann, Kolbe
  • Ethers: Williamson Synthesis, Cleavage with HI
  • Distinction Tests: Lucas, Iodoform, Victor Meyer

JEE Main Weightage

Typically 3-5 questions from this chapter. Focus on mechanisms, tests, preparations.

Weightage High (3-5 Qs)